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Design, Synthesis, and Anticancer Activity of Novel Trimethoxyphenyl-Derived Chalcone-Benzimidazolium Salts 期刊论文
ACS OMEGA, 2019, 卷号: 4, 期号: 23, 页码: 20381-20393
作者:  Yang, Jun-Li;  Ma, Yong-Hui;  Li, Yan-Hua;  Zhang, Yi-Peng;  Tian, Hong-Chang;  Huang, Yuan-Cheng;  Li, Yan;  Chen, Wen;  Yang, Li-Juan
浏览  |  Adobe PDF(2215Kb)  |  收藏  |  浏览/下载:302/57  |  提交时间:2020/03/18
Design and synthesis of novel artemisinin derivatives with potent activities against colorectal cancer in vitro and in vivo 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 182, 页码: 10
作者:  Wang, Liang-Liang;  Kong, Lingmei;  Liu, Hui;  Zhang, Yunqin;  Zhang, Li;  Liu, Xingyong;  Yuan, Feng;  Li, Yan;  Zuo, Zhili
收藏  |  浏览/下载:149/0  |  提交时间:2020/03/02
Artemisinin  Quinazoline  Hybridization  Colorectal cancer  Chemotherapy  
Alkaloids as Cyclooxygenase Inhibitors in Anticancer Drug Discovery 期刊论文
CURRENT PROTEIN & PEPTIDE SCIENCE, 2018, 卷号: 19, 期号: 3, 页码: 292-301
作者:  Hashmi, Muhammad Ali;  Khan, Afsar;  Farooq, Umar;  Khan, Sehroon
收藏  |  浏览/下载:105/0  |  提交时间:2018/05/08
Anticancer  Cyclooxygenase  Cox-2  Alkaloids  Enzyme Inhibition  Anti-inflammatory  Anti-tumor  
New phenolic glycosides from Curculigo orchioides and their xanthine oxidase inhibitory activities 期刊论文
FITOTERAPIA, 2017, 卷号: 122, 期号: 1, 页码: 144-149
作者:  Chen, Xinglong;  Zuo, Aixue;  Deng, Zhentao;  Huang, Xiaoyan;  Zhang, Xuemei;  Geng, Changan;  Li, Tianze;  Chen, Jijun
浏览  |  Adobe PDF(392Kb)  |  收藏  |  浏览/下载:261/75  |  提交时间:2017/12/18
Phenolic Glycosides  Xanthine Oxidase Inhibitory Activity  Curculigo Orchioides  
Synthesis and cytotoxic activity of novel hybrid compounds between 2-alkylbenzofuran and imidazole 期刊论文
MEDICINAL CHEMISTRY RESEARCH, 2014, 卷号: 23, 期号: 3, 页码: 1599-1611
作者:  Wan, Wei-Chao;  Chen, Wen;  Liu, Lan-Xiang;  Li, Yan;  Yang, Li-Juan;  Deng, Xiao-Yan;  Zhang, Hong-Bin;  Yang, Xiao-Dong
浏览  |  Adobe PDF(509Kb)  |  收藏  |  浏览/下载:825/536  |  提交时间:2014/04/09
Hybrid Compound  Benzofuran  Imidazole  Cytotoxic Activity  Structure-activity Relationships  Molecular Docking  
Pegaharmalines A and B, two novel beta-carboline alkaloids with unprecedented carbon skeletons from Peganum harmala 期刊论文
RSC ADVANCES, 2014, 卷号: 4, 期号: 96, 页码: 53725-53729
作者:  Wang, Kai-Bo;  Yuan, Chun-Mao;  Xue, Chun-Mei;  Li, Da-Hong;  Jing, Yong-Kui;  He, Hong-Ping;  Hao, Xiao-Jiang;  Di, Ying-Tong;  Li, Zhan-Lin;  Hua, Hui-Ming;  Hua,HM (reprint author),Shenyang Pharmaceut Univ,Key Lab Struct Based Drug Design & Discovery,Minist Educ,Shenyang 110016,Peoples R China.
浏览  |  Adobe PDF(585Kb)  |  收藏  |  浏览/下载:281/67  |  提交时间:2015/01/20
Liverwort Lepidolaena-clavigera  Caspase-3 Inhibitory-activity  Sp No 27  Absolute-configuration  Aspergillus-fumigatus  Tetracyclic Skeleton  Chaetomium-elatum  Phialophora  Metabolites  Acetals  
Design, synthesis and antitumor activity of novel 8-substituted 2,3,5,6-tetrahydrobenzo[1,2-b:4, 5-b'] difuran imidazolium salt derivatives 期刊论文
RSC ADVANCES, 2014, 卷号: 4, 期号: 31, 页码: 16312-16319
作者:  Sun, Cheng-Jun;  Chen, Wen;  Li, Yan;  Liu, Lan-Xiang;  Wang, Xue-Quan;  Li, Li-Juan;  Zhang, Hong-Bin;  Yang, Xiao-Dong
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Hybrid Compounds  Cytotoxic Activities  Natural-products  Drug Discovery  Analogs  Dihydrobenzofuran  Cycloaddition  Benzofurans  Iodides  Trans  
Asperterrestide A, a Cytotoxic Cyclic Tetrapeptide from the Marine-Derived Fungus Aspergillus terreus SCSGAF0162 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2013, 卷号: 76, 期号: 6, 页码: 1182-1186
作者:  He, Fei;  Bao, Jie;  Zhang, Xiao-Yong;  Tu, Zheng-Chao;  Shi, Yi-Ming;  Qi, Shu-Hua
浏览  |  Adobe PDF(237Kb)  |  收藏  |  浏览/下载:504/231  |  提交时间:2013/10/16
Cyanobacterium Lyngbya-majuscula  Metabolites  Biosynthesis  Derivatives  Agents  
Small-Molecule Inhibitors for the Treatment of Hepatitis B Virus Documented in Patents 期刊论文
MINI-REVIEWS IN MEDICINAL CHEMISTRY, 2013, 卷号: 13, 期号: 5, 页码: 749-776
作者:  Geng, Chang-An;  Wang, Li-Jun;  Guo, Rui-Hua;  Chen, Ji-Jun
浏览  |  Adobe PDF(616Kb)  |  收藏  |  浏览/下载:407/153  |  提交时间:2013/06/08
Hepatitis b Virus (Hbv)  Small-molecule Inhibitors  Nucleoside Analogs  Non-nucleosides  Natural Products  Synthesized Compounds  Chemical Modification  Patents  
Multicomplex-Based Pharmacophore-Guided 3D-QSAR Studies of N-Substituted 2'-(Aminoaryl)Benzothiazoles as Aurora-A Inhibitors 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2012, 卷号: 79, 期号: 6, 页码: 960-971
作者:  He, Gu;  Qiu, Minghua;  Li, Rui;  Ouyang, Liang;  Wu, Fengbo;  Song, Xiangrong;  Cheng, Li;  Xiang, Mingli;  Yu, Luoting
Adobe PDF(1377Kb)  |  收藏  |  浏览/下载:317/96  |  提交时间:2012/06/07
3d-qsar  Aurora-a  Kinase Inhibitors  Multicomplex-based Pharmacophore(Mcbp)  Pharmacophore