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The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP)1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-42
作者:  C Pergola;  J Gerstmeier;  B Monch;  B Çaliskan;  S Luderer;  C Weinige;  D Barz;  J Maczewsky;  S Pace;  A Rossi;  L Sautebin;  E Banoglu;  O Werz
Adobe PDF(1387Kb)  |  收藏  |  浏览/下载:483/1  |  提交时间:2017/07/24
Pharmacological characterizationof tachykinin tetrabranched derivatives 期刊论文
出版物, 3111, 期号: 0, 页码: 1-36
作者:  Chiara Ruzza;  Anna Rizzi;  Davide Malfacini;  Maria Camilla Cerlesi;  Federica Ferrari;  Erika Marzola;  Caterina Ambrosio;  Cristina Gro;  Salvadori Severo;  Tommaso Costa;  Girolamo Calo;  Remo Guerrini
Adobe PDF(1277Kb)  |  收藏  |  浏览/下载:300/1  |  提交时间:2017/07/24
Tachykinins  Substance p  Pwt2-sp  Nk1 Receptor  Calcium Mobilization  Bioluminescence Resonance Energy Transfer  Guinea Pig Ileum  Rat Urinary Bladder  Nociceptive Behaviour Induced By Spinal Substance p  Mice  
Structural and mechanistic basis of penicillin-bindingprotein inhibition by lactivicins 期刊论文
NATURE CHEMICAL BIOLOGY, 3111, 期号: 0, 页码: 1—5
作者:  Pauline Macheboeuf;  Delphine S Fischer;  Tom Brown Jr;  Astrid Zervosen;  Andre´Luxen;  Bernard Joris;  Andrea Dessen;  Christopher J Schofield
Adobe PDF(425Kb)  |  收藏  |  浏览/下载:251/1  |  提交时间:2017/07/21
Design and synthesis of guaianolide-germacranolide heterodimers as novel anticancer agents against hepatocellular carcinoma 期刊论文
DRUG DEVELOPMENT RESEARCH, 2023
作者:  Yan,Jia-Xin;  Li,Qi-Hao;  Li,Tian-Ze;  Huang,Zhi-Yan;  Ma,Yun-Bao;  Chen,Ji-Jun
浏览  |  Adobe PDF(7663Kb)  |  收藏  |  浏览/下载:169/33  |  提交时间:2024/07/10
antihepatoma effects  guaianolide-germacranolide heterodimers  PDGFRA  DERIVATIVES  
A new amide from the fruiting bodies of Tricholoma bakamatsutake 期刊论文
MAGNETIC RESONANCE IN CHEMISTRY, 2023, 卷号: 61, 期号: 7, 页码: 443-447
作者:  Zhang,Feng-Ming;  Lu,Bin;  Wang,Yue-Hu;  Yu,Fu-Qiang
浏览  |  Adobe PDF(380Kb)  |  收藏  |  浏览/下载:160/49  |  提交时间:2024/07/25
HONGO  
蕊木和奶子藤中生物碱类化学成分及其生物活性评价 学位论文
: 中国科学院大学, 2022
作者:  陈谌
Adobe PDF(17478Kb)  |  收藏  |  浏览/下载:731/1  |  提交时间:2024/05/14
夹竹桃科  Apocynaceae  蕊木  Kopsia arborea  奶子藤  Bousigonia mekongensis  单萜吲哚生物碱  Monoterterpene indole alkaloids  生物活性  Biological activity  
天然多糖AFG水凝胶的制备及其在皮肤创面愈合中的应用 学位论文
: 中国科学院大学, 2022
作者:  蒋泽秀
Adobe PDF(4884Kb)  |  收藏  |  浏览/下载:128/0  |  提交时间:2024/05/14
蜗牛糖胺聚糖,明胶,水凝胶,炎症,伤口愈合  Snail Glycosaminoglycan, Gelatin, Hydrogel, Inflammation, Wound Healing  
Pyranone Derivatives With Antitumor Activities, From the Endophytic Fungus Phoma sp. YN02-P-3 期刊论文
FRONTIERS IN CHEMISTRY, 2022, 卷号: 10, 页码: 950726
作者:  Yu, Chong;  Nian, Yin;  Chen, Huanhua;  Liang, Shuwen;  Sun, Mengyang;  Pei, Yuehu;  Wang, Haifeng
浏览  |  Adobe PDF(1148Kb)  |  收藏  |  浏览/下载:148/31  |  提交时间:2024/08/21
secondary metabolites  plant endophytic fungus  Phoma sp  pyranone derivatives  HL-60 inhibition  
Chemical constituents from plant endophytic fungus Alternaria alternata 期刊论文
NATURAL PRODUCT RESEARCH, 2021, 卷号: 35, 期号: 7, 页码: 1199-1206
作者:  Wang,Ju-Tao;  Ma,Zong-Hui;  Wang,Guo-Kai;  Xu,Feng-Qing;  Yu,Yang;  Wang,Gang;  Peng,Dai-Yin;  Liu,Jin-Song
收藏  |  浏览/下载:214/0  |  提交时间:2022/04/02
Alternaria alternata  Paeonia lactiflora  benzo-alpha-pyrone derivatives  cytotoxic activity  METABOLITES  INHIBITOR  ROOT  SP.  
Combined transcriptomic, proteomic and biochemical approaches to identify the cadmium hyper-tolerance mechanism of turnip seedling leaves 期刊论文
ENVIRONMENTAL SCIENCE AND POLLUTION RESEARCH, 2021, 卷号: 28, 期号: 18, 页码: 22458-22473
作者:  Li,Xiong;  Chen,Di;  Li,Boqun;  Yang,Ya;  Yang,Yongping
浏览  |  Adobe PDF(2377Kb)  |  收藏  |  浏览/下载:410/43  |  提交时间:2022/04/02
Turnip  Cadmium  Hyperaccumulator  Flavonoid  Acetylation  RNA-SEQ DATA  GENOME-WIDE IDENTIFICATION  GLUTATHIONE METABOLISM  SULFUR ASSIMILATION  GENE FAMILIES  STRESS  EFFLUX  ZINC  ACCUMULATION  PROTEIN