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The compound BTB06584 is an IF1-dependent selective inhibitor of the mitochondrial F1Fo-ATPase1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-38
作者:  Fabrice Ivanes;  Danilo Faccenda;  Jemma Gatliff;  Ahmed A Ahmed;  Stefania Cocco;  Carol Ho Ka Cheng;  Emma Allan;  Claire Russell;  Michael R Duchen;  Michelangelo Campanella
Adobe PDF(1228Kb)  |  收藏  |  浏览/下载:222/1  |  提交时间:2017/07/24
Mitochondrial F1fo Atp Synthase  If1  Ischemia-induced Death  Btb06584  Pinotage  
Effects of a new advanced glycation inhibitor, LR-90, on mitigating arterial stiffening and improving arterial elasticity and compliance in a diabetic rat model: aortic impedance analysis 期刊论文
出版物, 3111, 期号: 0, 页码: 1-33
作者:  S, Satheesan;  J L, Figarola;  T, Dabbs;  S, Rahbar;  R, Ermel
Adobe PDF(967Kb)  |  收藏  |  浏览/下载:258/1  |  提交时间:2017/07/24
Pharmacology and anti-addiction effects of the novel kappa opioid receptor agonist Mesyl Sal B, a potent and long-acting analogue of salvinorin A 期刊论文
出版物, 3111, 期号: 0, 页码: 1-53
作者:  B Simonson;  A S Morani;  A W M Ewald;  L Walker;  N Kumar;  D Simpson;  J H Miller;  T E Prisinzano;  B M Kivell
Adobe PDF(1394Kb)  |  收藏  |  浏览/下载:294/1  |  提交时间:2017/07/24
The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP)1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-42
作者:  C Pergola;  J Gerstmeier;  B Monch;  B Çaliskan;  S Luderer;  C Weinige;  D Barz;  J Maczewsky;  S Pace;  A Rossi;  L Sautebin;  E Banoglu;  O Werz
Adobe PDF(1387Kb)  |  收藏  |  浏览/下载:288/1  |  提交时间:2017/07/24
Pharmacological characterizationof tachykinin tetrabranched derivatives 期刊论文
出版物, 3111, 期号: 0, 页码: 1-36
作者:  Chiara Ruzza;  Anna Rizzi;  Davide Malfacini;  Maria Camilla Cerlesi;  Federica Ferrari;  Erika Marzola;  Caterina Ambrosio;  Cristina Gro;  Salvadori Severo;  Tommaso Costa;  Girolamo Calo;  Remo Guerrini
Adobe PDF(1277Kb)  |  收藏  |  浏览/下载:117/1  |  提交时间:2017/07/24
Tachykinins  Substance p  Pwt2-sp  Nk1 Receptor  Calcium Mobilization  Bioluminescence Resonance Energy Transfer  Guinea Pig Ileum  Rat Urinary Bladder  Nociceptive Behaviour Induced By Spinal Substance p  Mice  
The pharmacokinetics of anthocyanins and their metabolites in humans 期刊论文
出版物, 3111, 期号: 0, 页码: 1-37
作者:  R M de Ferrars;  C Czank;  Q Zhang;  N P Botting;  P A Kroon;  A Cassidy;  C D Kay
Adobe PDF(1873Kb)  |  收藏  |  浏览/下载:140/1  |  提交时间:2017/07/24
Anthocyanins  Metabolites  Hippuric Acid  Ferulic Acid  Vanillic Acid  
Resveratrol Decrease Fructose-Induced Oxidative Stress Mediated by NADPH Oxidase via an AMPK-Dependent Mechanism1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-44
作者:  Pei-Wen Cheng, PhD;  Wen-Yu Ho, MD, PhD;  Yu-Ting Su, MS;  Pei-Jung Lu,PhD;  Bo-Zone Chen MS;  Wen-Han Cheng, MS;  Wen-Hsien Lu, MD, MS;  Gwo-Ching Sun, MD;  Tung-Chen Yeh, MD;  Michael Hsiao DVM, PhD;  Ching-Jiunn Tseng, MD, PhD
Adobe PDF(1555Kb)  |  收藏  |  浏览/下载:129/1  |  提交时间:2017/07/24
Ampk  Hypertension  Nucleus Tractus Solitarii  Nitrogen Oxides  Resveratrol  
Nociceptin/Orphanin FQ peptide receptor antagonist JTC-801 reverses pain and anxiety symptoms in a rat model of PTSD 期刊论文
出版物, 3111, 期号: 0, 页码: 1-33
作者:  Y Zhang;  C D Simpson-Durand;  K M Standifer
Adobe PDF(1098Kb)  |  收藏  |  浏览/下载:127/1  |  提交时间:2017/07/24
中药砂仁降血糖活性成分研究 学位论文
: 中国科学院大学, 2022
作者:  丁敏
Adobe PDF(6349Kb)  |  收藏  |  浏览/下载:4/0  |  提交时间:2024/05/14
砂仁,姜科,降木脂素,降血糖活性,促GLP-1分泌,GPa抑制活性  Amomum villosum  Zingiberaceae  norlignans  antidiabetic effects  GLP-1 stimulation  GPa inhibition  
Hepatic RACK1 deletion disturbs lipid and glucose homeostasis independently of insulin resistance 期刊论文
JOURNAL OF ENDOCRINOLOGY, 2022, 卷号: 254, 期号: 3, 页码: 151-165
作者:  Qin, Wanying;  Zhang, Ting;  Ge, Mingxia;  Zhou, Huimin;  Xu, Yuhui;  Mu, Rongfang;  Huang, Chaoguang;  Liu, Daowei;  Huang, Bangrui;  Wang, Qian;  Kong, Qinghua;  Kong, Qingpeng;  Li, Fei;  Xiong, Wenyong
Adobe PDF(9525Kb)  |  收藏  |  浏览/下载:9/3  |  提交时间:2024/04/30
RACK1  bile acid  glucose metabolism  insulin sensitivity  ENDOPLASMIC-RETICULUM STRESS  C-KINASE 1  HEPATOCELLULAR-CARCINOMA  STEROL 12-ALPHA-HYDROXYLASE  DOWN-REGULATION  ER STRESS  KAPPA-B  RECEPTOR  ACTIVATION  GROWTH