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Synthesis and Cytotoxicity Evaluation of Tropinone Derivatives. 期刊论文
Natural products and bioprospecting, 2017, 卷号: 7, 期号: 2, 页码: 215-223
作者:  Yin, Xiu-Juan;  Geng, Chang-An;  Chen, Xing-Long;  Sun, Chang-Li;  Yang, Tong-Hua;  Li, Tian-Ze;  Zhou, Jun;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(758Kb)  |  收藏  |  浏览/下载:226/131  |  提交时间:2019/03/29
Bioactivity-guided synthesis of gramine derivatives as new MT1 and 5-HT1A receptors agonists 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2017, 卷号: 19, 期号: 6, 页码: 610-622
作者:  Yin, Xiu-Juan;  Huang, Xiao-Yan;  Ma, Yun-Bao;  Geng, Chang-An;  Li, Tian-Ze;  Chen, Xing-Long;  Yang, Tong-Hua;  Zhou, Jun;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(2718Kb)  |  收藏  |  浏览/下载:335/60  |  提交时间:2017/07/10
Gramine  Melatonin Receptor  5-hydroxy-tryptamine Receptor  Agonistic Activity  Structure-activity Relationships  
Bioactivity-guided synthesis of tropine derivatives as new agonists for melatonin receptors 期刊论文
RSC ADVANCES, 2016, 卷号: 6, 期号: 51, 页码: 45059-45063
作者:  Yin, Xiu-Juan;  Geng, Chang-An;  Huang, Xiao-Yan;  Chen, Hao;  Ma, Yun-Bao;  Chen, Xing-Long;  Sun, Chang-Li;  Yang, Tong-Hua;  Zhou, Jun;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(1380Kb)  |  收藏  |  浏览/下载:267/66  |  提交时间:2016/08/22
Synthesis and biological assay of 4-aryl-6-chloro-quinoline derivatives as novel non-nucleoside anti-HBV agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2011, 卷号: 19, 期号: 4, 页码: 1400-1408
作者:  Guo, Rui-Hua;  Zhang, Quan;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Luo, Jie;  Wang, Li-Jun;  Geng, Chang-An;  Zhang, Xue-Mei;  Zhou, Jun;  Jiang, Zhi-Yong;  Chen, Ji-Jun
Adobe PDF(951Kb)  |  收藏  |  浏览/下载:459/145  |  提交时间:2012/04/10
Hepatitis b Virus  4-aryl-6-chloro-quinoline  Derivatives  Synthesis  
Structure-activity relationships study of 6-chloro-4-(2-chlorophenyl)-3-(2-hydroxyethyl) quinolin-2(1H)-one derivatives as novel non-nucleoside anti-hepatitis B virus agents 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2011, 卷号: 46, 期号: 1, 页码: 307-319
作者:  Guo, Rui-Hua;  Zhang, Quan;  Ma, Yun-Bao;  Luo, Jie;  Geng, Chang-An;  Wang, Li-Jun;  Zhang, Xue-Mei;  Zhou, Jun;  Jiang, Zhi-Yong;  Chen, Ji-Jun
Adobe PDF(866Kb)  |  收藏  |  浏览/下载:358/91  |  提交时间:2012/04/10
Anti-hepatitis b Virus Activity  Quinolin-2(1h)-one  Structure-activity Relationships  
Anti-HBV agents. Part 3: Preliminary structure-activity relationships of tetra-acylalisol A derivatives as potent hepatitis B virus inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 卷号: 19, 期号: 23, 页码: 6659-6665
作者:  Zhang, Quan;  Jiang, Zhi-Yong;  Luo, Jie;  Ma, Yun-Bao;  Liu, Ji-Feng;  Guo, Rui-Hua;  Zhang, Xue-Mei;  Zhou, Jun;  Niu, Wei;  Du, Fei-Fei;  Li, Li;  Li, Chuan;  Chen, Ji-Jun
Adobe PDF(2076Kb)  |  收藏  |  浏览/下载:499/130  |  提交时间:2012/03/21
Anti-hbv Activity  Protostane-type Triterpene  Alisol a  Derivatives  Chemical Modification  
Anti-HBV agents. Part 2: Synthesis and in vitro anti-hepatitis B virus activities of alisol A derivatives 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 卷号: 19, 期号: 8, 页码: 2148-2153
作者:  Zhang, Quan;  Jiang, Zhi-Yong;  Luo, Jie;  Liu, Ji-Feng;  Ma, Yun-Bao;  Guo, Rui-Hua;  Zhang, Xue-Mei;  Zhou, Jun;  Chen, Ji-Jun
Adobe PDF(2279Kb)  |  收藏  |  浏览/下载:364/112  |  提交时间:2011/12/19
Anti-hbv Activity  Protostane-type Triterpene  Alisol a  Derivatives  Chemical Modification  
Anti-HBV agents. Part 1: Synthesis of alisol A derivatives: A new class of hepatitis B virus inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 卷号: 18, 期号: 16, 页码: 4647-4650
作者:  Zhang, Quan;  Jiang, Zhi-Yong;  Luo, Jie;  Cheng, Pi;  Ma, Yun-Bao;  Zhang, Xue-Mei;  Zhang, Feng-Xue;  Zhou, Jun;  Chen, Ji-Jun
Adobe PDF(173Kb)  |  收藏  |  浏览/下载:255/79  |  提交时间:2011/11/24
Anti-hbv Activity  Alisol a  Derivatives  Synthesis  
Synthesis and biological evaluation of N-acetyl-beta-aryl-1,2-didehydroethylamines as new HIV-1 RT inhibitors in vitro 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 卷号: 17, 期号: 16, 页码: 4476-4480
作者:  Cheng, Pi;  Jiang, Zhi-Yong;  Wang, Rul-Rul;  Zhang, Xue-Mel;  Wang, Qian;  Zheng, Yong-Tang;  Zhou, Jun;  Chen, Ji-Jun
Adobe PDF(148Kb)  |  收藏  |  浏览/下载:359/112  |  提交时间:2011/11/24
Beta-aryl-nitroolefin  N-acetyl-beta-aryl-1  Nnrtis  2-didehydroethylamine  Anti-hiv-1 Rt Activity