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Design, synthesis and structure-activity relationship optimization of phenanthridine derivatives as new Wnt/beta-catenin signalling pathway agonists 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 84, 页码: 285-294
作者:  Chen, Duo-zhi;  Yang, Bi-juan;  He, Xiao-li;  Fan, Shi-rui;  Cai, Jie-yun;  Jing, Chen-xu;  Zhang, Heng;  Zhang, Yu;  Li, Lin;  Hao, Xiao-jiang
浏览  |  Adobe PDF(3047Kb)  |  收藏  |  浏览/下载:285/35  |  提交时间:2019/03/18
Wnt/beta-catenin signalling pathway agonist  Phenanthridine derivatives  Structural optimization  Structure-activity relationships (SARs)  
Synthesis of Novel ent-Kaurane-Type Diterpenoid Derivatives Effective for Highly Aggressive Tumor Cells 期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 12, 页码: 9
作者:  Hu, Yu;  Li, Xiao-Nian;  Ma, Ze-Jin;  Puno, Pema-Tenzin;  Zhao, Yong;  Zhao, Yan;  Xiao, Ye-Zhi;  Zhang, Wei;  Liu, Jing-Ping
收藏  |  浏览/下载:121/0  |  提交时间:2019/03/18
ent-kaurane-type diterpenoid derivatives  antitumor  synthesis  
New phloroglucinol derivatives with protein tyrosine phosphatase 1B (PTP1B) inhibitory activities from Syzygium austroyunnanense 期刊论文
FITOTERAPIA, 2018, 卷号: 131, 页码: 141-145
作者:  Xu, Shao-Hua;  Xu, Wen;  Wang, Li;  Hu, Yi-Kao;  Liu, Jin-Ping;  Zhao, Yan;  Li, Meng-Jia;  Li, Feng;  Huang, Sheng-Xiong;  Zhao, Yong
收藏  |  浏览/下载:112/0  |  提交时间:2019/03/18
Syzygium austroyunnanense  Myrtaceae  Phloroglucinol derivatives  Structure elucidation  PTP 1B inhibitory activities  
Efficient synthesis of new phenanthridine Wnt/beta-catenin signaling pathway agonists 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 157, 页码: 1491-1499
作者:  Chen, Duozhi;  Zhang, Heng;  Jing, Chenxu;  He, Xiaoli;  Yang, Bijuan;  Cai, Jieyun;  Zhou, Yunfu;  Song, Xiaoming;  Li, Lin;  Hao, Xiaojiang
收藏  |  浏览/下载:350/0  |  提交时间:2018/11/12
Wnt/beta-catenin signaling agonist  Phenanthridine derivatives  Structural optimization  
Synthesis and biological evaluation of magnolol derivatives as melatonergic receptor agonists with potential use in depression 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 期号: 0, 页码: 381-393
作者:  Yang, Tong-Hua;  Ma, Yun-Bao;  Geng, Chang-An;  Yan, De-Xiu;  Huang, Xiao-Yan;  Li, Tian-Ze;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(2088Kb)  |  收藏  |  浏览/下载:197/68  |  提交时间:2018/10/04
Depression  Magnolol Derivatives  Mt1/2 Receptors  Metabolites  Monoamine Neurotransmitter  
Cytotoxicity-Guided Isolation of Two New Phenolic Derivatives from Dryopteris fragrans (L.) Schott 期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 7, 页码: 11
作者:  Zhang, Tong;  Wang, Li;  Duan, De-Hua;  Zhang, Yi-Hao;  Huang, Sheng-Xiong;  Chang, Ying
收藏  |  浏览/下载:115/0  |  提交时间:2018/11/12
cytotoxicity-guided  phenolic derivatives  Dryopteris fragrans  chemical derivatization  immuno-regulation activity