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Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:360/39  |  提交时间:2017/12/18
Polycyclic Azetidines and Pyrrolidines via Palladium-Catalyzed Intramolecular Amination of Unactivated C(sp3)-H Bonds 期刊论文
ORGANIC LETTERS, 2017, 卷号: 19, 期号: 18, 页码: 4880-4883
作者:  Zhao, Jie;  Zhao, Xiao-Jing;  Cao, Pei;  Liu, Ji-Kai;  Wu, Bin
Adobe PDF(1162Kb)  |  收藏  |  浏览/下载:211/60  |  提交时间:2017/10/23
C-h Functionalization  c(Sp(3))-h Bonds  Beta-lactams  Stereoselective-synthesis  Organic-synthesis  Aliphatic-amines  Activation  Derivatives  Cyclization  Amidation  
Click Glycosylation for the Synthesis of 1,2,3-Triazole-Linked Picropodophyllotoxin Glycoconjugates and Their Anticancer Activity 期刊论文
CHEMISTRYSELECT, 2017, 卷号: 2, 期号: 18, 页码: 5038-5044
作者:  Zi, Cheng-Ting;  Yang, Liu;  Gao, Wei;  Li, Yan;  Zhou, Jun;  Ding, Zhong-Tao;  Hu, Jiang-Miao;  Jiang, Zi-Hua
Adobe PDF(3775Kb)  |  收藏  |  浏览/下载:206/42  |  提交时间:2017/10/23
Anticancer Activity  Cu(i)-catalyzed Click Reaction  Glycoconjugates  Picropodophyllotoxin  Podophyllotoxin  
Discovery of new dual binding TNKS inhibitors of Wnt signaling inhibition by pharmacophore modeling, molecular docking and bioassay 期刊论文
MOLECULAR BIOSYSTEMS, 2017, 卷号: 13, 期号: 2, 页码: 363-370
作者:  Pu, Yinglan;  Zhang, Shuqun;  Chang, Zhe;  Zhang, Yunqin;  Wang, Dong;  Zhang, Li;  Li, Yan;  Zuo, Zhili
Adobe PDF(972Kb)  |  收藏  |  浏览/下载:659/116  |  提交时间:2017/05/19