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UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations Eph antagonist and angiogenesis 期刊论文
出版物, 3111, 期号: 0, 页码: 1-32
Authors:  I Hassan-Mohamed;  C Giorgio;  M Incerti;  S Russo;  D Pala;  E B Pasquale;  P Vicini;  E Barocelli;  S Rivara;  M Mor;  A Lodola;  M Tognolini
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Eph Kinase  Ephrin  Small Molecules  Angiogenesis  Bile Acid  Lithocholic Acid  
The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP)1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-42
Authors:  C Pergola;  J Gerstmeier;  B Monch;  B Çaliskan;  S Luderer;  C Weinige;  D Barz;  J Maczewsky;  S Pace;  A Rossi;  L Sautebin;  E Banoglu;  O Werz
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Structural and mechanistic basis of penicillin-bindingprotein inhibition by lactivicins 期刊论文
NATURE CHEMICAL BIOLOGY, 3111, 期号: 0, 页码: 1—5
Authors:  Pauline Macheboeuf;  Delphine S Fischer;  Tom Brown Jr;  Astrid Zervosen;  Andre´Luxen;  Bernard Joris;  Andrea Dessen;  Christopher J Schofield
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YC-1 inhibits proliferation of breast cancer cells by downregulating EZH2 expression via activation of c-Cbl and ERK 期刊论文
出版物, 3111, 期号: 0, 页码: 1-46
Authors:  Ling-Chu Chang;  Hui-Yi Lin;  Meng-Tung Tsai;  Ruey-Hwang Chou;  Fang-Yu Lee;  Che-Ming Teng;  Min-Tsang Hsieh;  Hsin-Yi Hung;  Li-Jiau Huang;  Yung-Luen Yu;  Sheng-Chu Kuo
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Yc-1  Triple-negative Breast Cancer  Erk  Ezh2  C-cbl  
Antidepressant and anxiolytic profiles of newly synthesized arginine vasopressin 期刊论文
出版物, 3111, 期号: 0, 页码: 1-62
Authors:  M Iijima;  T Yoshimizu;  T Shimazaki;  K Tokugawa;  K Fukumoto;  S Kurosu;  T Kuwada;  Y Sekiguchi;  S Chaki
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Arginine Vasopressin  V1b Receptor Antagonist  Depression  Anxiety  Hpa Axis  
Nociceptin/Orphanin FQ peptide receptor antagonist JTC-801 reverses pain and anxiety symptoms in a rat model of PTSD 期刊论文
出版物, 3111, 期号: 0, 页码: 1-33
Authors:  Y Zhang;  C D Simpson-Durand;  K M Standifer
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The Tyrosine Kinase Inhibitor Bafetinib Inhibits PAR2-induced Activation of TRPV4 In Vitro and Pain In Vivo1 期刊论文
出版物, 2111, 页码: 1-44
Authors:  1M S Grace;  T Lieu;  B Darby;  F C Abogadie;  N Veldhuis N W Bunnett;  P McIntyre
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Transient Receptor Potential Ion Channel  Trpv4  Protease Activated Receptor  Par2  Pain  Tyrosine Kinase  Bafetinib  
Synthesis and biological evaluation of novel 3-benzylcoumarin-imidazolium salts 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 4, 页码: 6
Authors:  Wang, Xue-Quan;  Chen, Xue-Bing;  Ye, Ping-Ting;  Yang, Zhi-Xin;  Bai, Meng-Jiao;  Duan, Su-Yue;  Li, Yan;  Yang, Xiao-Dong
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3-Benzylcoumarin  Imidazolium salts  Biological evaluation  Cytotoxic activity  Structure-activity relationships  
Phyllanthacidoid U: a new N-glycosyl norbisabolane sesquiterpene from Phyllanthus acidus (L.) skeels 期刊论文
NATURAL PRODUCT RESEARCH, 2020, 页码: 8
Authors:  Xin, Ying;  Xu, Min;  Wang, Ya-Feng;  Zheng, Xiao-Hong;  Zhu, Hong-Tao;  Wang, Dong;  Yang, Chong-Ren;  Zhang, Ying-Jun
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Phyllanthus acidus  phyllanthacidoid U  norbisabolane sesquiterpenoid  amide  
Benwamycins A-G, Trialkyl-Substituted Benzene Derivatives from a Soil-Derived Streptomyces 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2020, 卷号: 83, 期号: 1, 页码: 111-117
Authors:  Yang, Feng-Xian;  Huang, Jian-Ping;  Liu, Zhixiang;  Wang, Zhiyan;  Yang, Jing;  Tang, Jun;  Yu, Zhiyin;  Yan, Yijun;  Kai, Guoyin;  Huang, Sheng-Xiong
Favorite  |  View/Download:67/0  |  Submit date:2020/03/24