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UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations Eph antagonist and angiogenesis 期刊论文
出版物, 3111, 期号: 0, 页码: 1-32
作者:  I Hassan-Mohamed;  C Giorgio;  M Incerti;  S Russo;  D Pala;  E B Pasquale;  P Vicini;  E Barocelli;  S Rivara;  M Mor;  A Lodola;  M Tognolini
Adobe PDF(1403Kb)  |  收藏  |  浏览/下载:235/1  |  提交时间:2017/07/24
Eph Kinase  Ephrin  Small Molecules  Angiogenesis  Bile Acid  Lithocholic Acid  
分子模拟应用于岩藻糖化糖胺聚糖 3D 结构确定及其与内源 性因子 X 酶的相互作用模式考察 学位论文
, 2021
作者:  陈鼎元
Adobe PDF(4948Kb)  |  收藏  |  浏览/下载:39/0  |  提交时间:2023/11/02
Vincan- and eburnan-type alkaloids from Tabernaemontana bovina and their hypoglycemic activity 期刊论文
PHYTOCHEMISTRY, 2021, 卷号: 190, 页码: 112859
作者:  Yu,Yang;  Bao,Mei-Fen;  Huang,Sheng-Zhuo;  Wu,Jing;  Cai,Xiang-Hai
浏览  |  Adobe PDF(5274Kb)  |  收藏  |  浏览/下载:89/44  |  提交时间:2022/04/02
Tabernaemontana bovina  Apocynaceae  Vincan-type alkaloids  Eburnan-type alkaloids  Hypoglycemic activity  INDOLE ALKALOIDS  
A non-anticoagulant heparin-like snail glycosaminoglycan promotes healing of diabetic wound 期刊论文
CARBOHYDRATE POLYMERS, 2020
作者:  Wu, Yuebo;  Zhou, Zhipeng;  Luo, Lan;  Tao, Maixian;  Chang, Xiao;  Yang, Lian;  Huang, Xingyong;  Hu, Lin;  Wu, Mingyi
浏览  |  Adobe PDF(3690Kb)  |  收藏  |  浏览/下载:73/32  |  提交时间:2021/01/05
Rhodamine B-based fluorescent probes for molecular mechanism study of the anti-influenza activity of pentacyclic triterpenes 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020
作者:  Li, Man;  Yuan, Lan;  Chen, Yingying;  Ma, Wenxiao;  Ran, Fuxiang;  Zhang, Lihe;  Zhou, Demin;  Xiao, Sulong
浏览  |  Adobe PDF(2312Kb)  |  收藏  |  浏览/下载:85/29  |  提交时间:2021/01/05
Discovery of highly functionalized 5,6-seco-grayanane diterpenoids as potent competitive PTP1B inhibitors 期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2020
作者:  Zhou, Junfei;  Zuo, Zhili;  Liu, Junjun;  Zhang, Hanqi;  Zheng, Guijuan;  Yao, Guangmin
浏览  |  Adobe PDF(1539Kb)  |  收藏  |  浏览/下载:102/21  |  提交时间:2021/01/05
Dalbavancin binds ACE2 to block its interaction with SARS-CoV-2 spike protein and is effective in inhibiting SARS-CoV-2 infection in animal models 期刊论文
CELL RESEARCH, 2020
作者:  Wang, Gan;  Yang, Meng-Li;  Duan, Zi-Lei;  Liu, Feng-Liang;  Jin, Lin;  Long, Cheng-Bo;  Zhang, Min;  Tang, Xiao-Peng;  Xu, Ling;  Li, Ying-Chang;  Kamau, Peter Muiruri;  Yang, Lian;  Liu, Hong-Qi;  Xu, Jing-Wen;  Chen, Jie-Kai;  Zheng, Yong-Tang;  Peng, Xiao-Zhong;  Lai, Ren
浏览  |  Adobe PDF(2926Kb)  |  收藏  |  浏览/下载:99/33  |  提交时间:2021/01/05
Identification and Characterization of ShSPI, a Kazal-Type Elastase Inhibitor from the Venom of Scolopendra Hainanum 期刊论文
TOXINS, 2019, 卷号: 11, 期号: 12, 页码: 13
作者:  Luan, Ning;  Zhao, Qiyu;  Duan, Zilei;  Ji, Mengyao;  Xing, Meichen;  Zhu, Tengyu;  Mwangi, James;  Rong, Mingqiang;  Liu, Jiangxin;  Lai, Ren
浏览  |  Adobe PDF(2415Kb)  |  收藏  |  浏览/下载:132/28  |  提交时间:2020/03/18
centipede  kazal-type inhibitor  human neutrophils elastase  ShSPI  
Nonasaccharide Inhibits Intrinsic Factor Xase Complex by Binding to Factor IXa and Disrupting Factor IXa-Factor VIIIa Interactions 期刊论文
THROMBOSIS AND HAEMOSTASIS, 2019, 卷号: 119, 期号: 5, 页码: 705-715
作者:  Xiao, Chuang;  Zhao, Longyan;  Gao, Na;  Wu, Mingyi;  Zhao, Jinhua
浏览  |  Adobe PDF(740Kb)  |  收藏  |  浏览/下载:186/49  |  提交时间:2019/06/24
nonasaccharide from fucosylated glycosaminoglycan  intrinsic factor Xase complex  factor IXa  anticoagulant  
Microbe-focused glycan array screening platform 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2019, 卷号: 116, 期号: 6, 页码: 1958-1967
作者:  Geissner, Andreas;  Reinhardt, Anika;  Rademacher, Christoph;  Johannssen, Timo;  Monteiro, Joao;  Lepenies, Bernd;  Thepaut, Michel;  Fieschi, Franck;  Mrazkova, Jana;  Wimmerova, Michaela;  Schuhmacher, Frank;  Goetze, Sebastian;  Gruenstein, Dan;  Guo, Xiaoqiang;  Hahm, Heung Sik;  Kandasamy, Jeyakumar;  Leonori, Daniele;  Martin, Christopher E.;  Parameswarappa, Sharavathi G.;  Pasari, Sandip;  Schlegel, Mark K.;  Tanaka, Hidenori;  Xiao, Guozhi;  Yang, You;  Pereira, Claney L.;  Anish, Chakkumkal;  Seeberger, Peter H.
浏览  |  Adobe PDF(1198Kb)  |  收藏  |  浏览/下载:187/33  |  提交时间:2019/03/18
glycan arrays  microbial antigens  immune receptors  antiglycan antibodies  bacterial lectins