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Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:408/46  |  提交时间:2017/12/18
Identification and validation of p50 as the cellular target of eriocalyxin B 期刊论文
ONCOTARGET, 2014, 卷号: 5, 期号: 22, 页码: 11354-11364
作者:  Kong, Ling-Mei;  Deng, Xu;  Zuo, Zhi-Li;  Sun, Han-Dong;  Zhao, Qin-Shi;  Li, Yan
浏览  |  Adobe PDF(3014Kb)  |  收藏  |  浏览/下载:319/80  |  提交时间:2015/06/17
Erib  Activity-based Probes  P50  Nf-kappa b Signaling  Apoptosis  
Dual-Functional abeo-Taxane Derivatives Destabilizing Microtubule Equilibrium and Inhibiting NF-kappa B Activation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 11, 页码: 4749-4757
作者:  Zhao, Yu;  Su, Jia;  Goto, Masuo;  Morris-Natschke, Susan L.;  Li, Yan;  Zhao, Qin-Shi;  Yao, Zhu-Jun;  Lee, Kuo-Hsiung
浏览  |  Adobe PDF(531Kb)  |  收藏  |  浏览/下载:346/82  |  提交时间:2013/10/16
Natural-products  Biological-activity  Cancer-therapy  Paclitaxel  Taxol  Resistance  Drugs  Chemotherapy  Parthenolide  Brevifoliol  
Norditerpenoids from Salvia castanea Diels f. pubescens 期刊论文
FITOTERAPIA, 2012, 卷号: 83, 期号: 6, 页码: 1072-1075
作者:  Pan, Zheng-Hong;  Li, Yan;  Wu, Xing-De;  He, Juan;  Chen, Xuan-Qin;  Xu, Gang;  Peng, Li-Yan;  Zhao, Qin-Shi
浏览  |  Adobe PDF(278Kb)  |  收藏  |  浏览/下载:612/187  |  提交时间:2012/11/30
Salvia Castanea Diels F. Pubescens  Norditerpenoid  Castanol A-c  Cytotoxic Activity  
Development of novel conformation-constrained cytotoxic derivatives of cheliensisin A by embedment of small heterocycles 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2011, 卷号: 46, 期号: 9, 页码: 4238-4244
作者:  Deng, Xu;  Su, Jia;  Zhao, Yu;  Peng, Li-Yan;  Li, Yan;  Yao, Zhu-Jun;  Zhao, Qin-Shi
Adobe PDF(450Kb)  |  收藏  |  浏览/下载:413/103  |  提交时间:2012/03/16
Cheliensisin a  Derivative  Structure-activity Relationship  Cytotoxicity  Anticancer  
Diterpenoid Constituents of the Roots of Salvia digitaloides 期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2010, 卷号: 58, 期号: 23, 页码: 12157-12161
作者:  Xu, Gang;  Yang, Jing;  Wang, Yuan-Yuan;  Peng, Li-Yan;  Yang, Xian-Wen;  Pan, Zheng-Hong;  Liu, En-De;  Li, Yan;  Zhao, Qin-Shi
Adobe PDF(839Kb)  |  收藏  |  浏览/下载:423/145  |  提交时间:2012/03/21
Salvia Digitaloides  Cytotoxic Activity  Diterpenoids  Stereochemistry