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中国科学院昆明植物研究所知识管理系统
Knowledge Management System of Kunming Institute of Botany,CAS
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Celastrol as an intestinal FXR inhibitor triggers tripolide-induced intestinal bleeding: Underlying mechanism of gastrointestinal injury induced by Tripterygium wilfordii
期刊论文
PHYTOMEDICINE, 2023, 卷号: 121, 页码: 155054
作者:
Dai,Manyun
;
Peng,Wan
;
Lin,Lisha
;
Wu,Zhanxuan
;
Zhang,Ting
;
Zhao,Qi
;
Cheng,Yan
;
Lin,Qiuxia
;
Zhang,Binbin
;
Liu,Aiming
;
Rao,Qianru
;
Huang,Jianfeng
;
Zhao,Jinhua
;
Gonzalez,Frank J.
;
Li,Fei
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浏览/下载:28/18
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提交时间:2024/07/17
Intestinal bleeding
Triptolide
Celastrol
Intestinal FXR
Tripterygium wilfordii
FARNESOID-X-RECEPTOR
BACTERIAL TRANSLOCATION
ACTIVATION
INFLAMMATION
DYSFUNCTION
TRIPTOLIDE
MICROBIOTA
PREVENTS
OBESITY
MICE
Rubiginosin B selectively inhibits Treg cell differentiation and enhances anti-tumor immune responses by targeting calcineurin-NFAT signaling pathway
期刊论文
PHYTOMEDICINE, 2023, 卷号: 116, 页码: 154898
作者:
Geng,Chang-An
;
Chen,Feng-Yang
;
Zheng,Jing-Bin
;
Liao,Ping
;
Li,Tian-Ze
;
Zhang,Xue-Mei
;
Chen,Xin
;
Chen,Ji-Jun
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浏览/下载:28/10
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提交时间:2024/07/17
Rubiginosin B (RGB)
CD4(+)Foxp3(+) regulatory T cells (Tregs)
Calcineurin
Nuclear factor of activated T cells (NFAT)
Tumor microenvironment
Rhododendron brachypodum
REGULATORY T-CELLS
RHODODENDRON
IMMUNOSUPPRESSION
DERIVATIVES
INDUCTION
EXPANSION
RAPAMYCIN
Rearranged Homoadamantane-Type Polycyclic Polyprenylated Acylphloroglucinols from Hypericum pseudohenryi
期刊论文
ORGANIC LETTERS, 2023, 卷号: 25, 期号: 50, 页码: 8965-8969
作者:
Jiang,Na-Na
;
Ye,Yan-Song
;
Liu,Xia
;
Wang,Yong-Ling
;
Xu,Gang
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浏览/下载:17/6
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提交时间:2024/07/10
Identification of New Diterpenoids from the Pulp of Coffea arabica and Their α-Glucosidase Inhibition Activity
期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2023, 卷号: 72, 期号: 3, 页码: 1683-1694
作者:
Al-Romaima,Abdulbaset
;
Hu,Guilin
;
Wang,Yanbing
;
Quan,Chenxi
;
Dai,Haopeng
;
Qiu,Minghua
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浏览/下载:27/12
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提交时间:2024/07/10
Coffeaarabica
coffee pulp
diterpenoids
structure elucidation
alpha-glucosidase
moleculardocking
ENT-KAURANE DITERPENES
ACID
PRODUCTS
EXTRACTS
CAFFEINE
CAFESTOL
ESTERS
BEANS
Discovery of potential novel TRPC5 inhibitors by virtual screening and bioassay
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 94, 页码: 117477
作者:
Shen,Meiling
;
Li,Lingfeng
;
Li,Yue
;
Gu,Xi
;
Bai,Longhui
;
Xia,Chengfeng
;
Xiong,Wenyong
;
Zuo,Zhili
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Adobe PDF(6089Kb)
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浏览/下载:25/8
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提交时间:2024/07/22
TRPC5
Inhibitors
Virtual screening
Ca 2+channel
CHANNELS
IDENTIFICATION
PERMEABILITY
CALCIUM
Discovery of 2-(Methylcarbonylamino) thiazole as PDE4 inhibitors via virtual screening and biological evaluation
期刊论文
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2023, 卷号: 124, 页码: 108567
作者:
Ma,Rui
;
Song,Na
;
Wang,Lveli
;
Gu,Xi
;
Xiong,Feng
;
Zhang,Shuqun
;
Zhang,Jie
;
Yang,Weimin
;
Zuo,Zhili
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Adobe PDF(5778Kb)
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浏览/下载:20/10
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提交时间:2024/07/22
PHOSPHODIESTERASE-4 INHIBITOR
ACCURATE DOCKING
APREMILAST
EFFICACY
INSIGHTS
DISEASE
ASTHMA
POTENT
GLIDE
Bioassay-guided isolation of α-Glucosidase inhibitory constituents from Hypericum sampsonii
期刊论文
CHINESE JOURNAL OF NATURAL MEDICINES, 2023, 卷号: 21, 期号: 6, 页码: 443-453
作者:
Tao,Linlan
;
Xu,Shuangyu
;
Zhang,Zizhen
;
Li,Yanan
;
Yang,Jue
;
Gu,Wei
;
Yi,Ping
;
Hao,Xiaojiang
;
Yuan,Chunmao
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Adobe PDF(1033Kb)
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浏览/下载:23/10
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提交时间:2024/07/22
Hypericum sampsonii
Chemical constituents
Structure elucidation
alpha-Glucosidase
Molecular docking
POLYCYCLIC POLYPRENYLATED ACYLPHLOROGLUCINOLS
POTENT INHIBITORS
SPECTROSCOPY
DERIVATIVES
CHEMISTRY
AMYLASE
ROOTS
Oligomeric phloroglucinols with hAChE inhibitory and antibacterial activities from tropic Rhodomyrtus tomentosa
期刊论文
BIOORGANIC CHEMISTRY, 2023, 卷号: 141, 页码: 106836
作者:
Luo,E-E
;
Liu,Si-Na
;
Wang,Zhao-Jie
;
Chen,Ling-Yun
;
Liang,Cheng-Qin
;
Yu,Mu-Yuan
;
Qin,Xu-Jie
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Adobe PDF(3972Kb)
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浏览/下载:21/8
  |  
提交时间:2024/07/22
Rhodomyrtus tomentosa
Oligomeric phloroglucinols
h AChE inhibitors
Molecular docking
Antibacterial effects
MYRTUCOMMULONE
DERIVATIVES
ACYLPHLOROGLUCINOLS
MYRTUCOMMUACETALONE
LEAVES
Artemiprinolides A-M, thirteen undescribed sesquiterpenoid dimers from Artemisia princeps and their antihepatoma activity
期刊论文
PHYTOCHEMISTRY, 2023, 卷号: 211, 页码: 113714
作者:
Su,Li-Hua
;
Ma,Wen-Jing
;
Ma,Yun-Bao
;
Li,Tian-Ze
;
Geng,Chang-An
;
Dong,Wei
;
He,Xiao-Feng
;
Chen,Ji-Jun
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Adobe PDF(7208Kb)
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浏览/下载:30/18
  |  
提交时间:2024/07/22
Artemisia princeps Pamp
Sesquiterpenoid dimers
Artemiprinolides A-M
Antihepatoma activity
Apoptosis
FARNESYL-PROTEIN TRANSFERASE
ETHANOL EXTRACT
PAMPANINI
INHIBITORS
JACEOSIDIN
Structurally modified Cyclovirobuxine-D Buxus alkaloids as effective analgesic agents through Cav3.2 T-Type calcium channel inhibition
期刊论文
BIOORGANIC CHEMISTRY, 2023, 卷号: 135, 页码: 106493
作者:
Munikishore,Rachakunta
;
Liu,Rui
;
Zhang,Shuqun
;
Zhao,Qin-Shi
;
Nian,Yin
;
Zuo,Zhili
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Adobe PDF(5035Kb)
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浏览/下载:27/5
  |  
提交时间:2024/07/22
Buxus alkaloid
Structural modification
T -type calcium channel
Analgesic activity
Docking analysis
Structure -activity relationship study
BUXOZINE-C
SEMPERVIRENS
RING
CONSTITUTION