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先导化合物设计与开发 学位论文
: 中国科学院大学, 2022
作者:  Munikishore Rachakunta
Microsoft Word(14465Kb)  |  收藏  |  浏览/下载:25/0  |  提交时间:2024/05/14
Buxus alkaloids  Buxus alkaloids  Cyclovirobuxine-D  Cyclovirobuxine-D  Synthesis, Calcium channel inhibitors  Synthesis, Calcium channel inhibitors  SAR studies  SAR studies  Anti-cardiovascular agents.  Anti-cardiovascular agents.  
Cyclovirobuxine D, a cardiovascular drug from traditional Chinese medicine, alleviates inflammatory and neuropathic pain mainly via inhibition of voltage-gated Ca(v)3.2 channels 期刊论文
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 1081697
作者:  Su, Deyuan;  Gong, Ye;  Li, Songyu;  Yang, Jian;  Nian, Yin
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Cyclovirobuxine D  Ca(v)3  2  Ca(v)2  Buxus microphylla  analgesic effects  ROOT GANGLION NEURONS  CALCIUM-CHANNELS  CELL-PROLIFERATION  PACLITAXEL  RAT  RECEPTOR  GENE  EXPRESSION  APOPTOSIS  CURRENTS