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Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:408/46  |  提交时间:2017/12/18
Two novel diterpenoid heterodimers, Bisebracteolasins A and B, from Euphorbia ebracteolata Hayata, and the cancer chemotherapeutic potential of Bisebracteolasin A 期刊论文
SCIENTIFIC REPORTS, 2017, 卷号: 7, 页码: 1
作者:  Yuan, Wen-Juan;  Ding, Xiao;  Wang, Zhe;  Yang, Bi-Juan;  Li, Xiao-Nian;  Zhang, Yu;  Chen, Duo-Zhi;  Li, Shun-Lin;  Chen, Quan;  Di, Ying-Tong;  Aisa, Haji Akber;  Hao, Xiao-Jiang
浏览  |  Adobe PDF(3375Kb)  |  收藏  |  浏览/下载:315/63  |  提交时间:2017/12/18
Natural Cyclopeptide RA-XII, a New Autophagy Inhibitor, Suppresses Protective Autophagy for Enhancing Apoptosis through AMPK/mTOR/P70S6K Pathways in HepG2 Cells 期刊论文
MOLECULES, 2017, 卷号: 22, 期号: 11, 页码: UNSP 1934
作者:  Song, Lihua;  Wang, Zhe;  Wang, Yurong;  Guo, Di;  Yang, Jianhong;  Chen, Lijuan;  Tan, Ninghua
浏览  |  Adobe PDF(4110Kb)  |  收藏  |  浏览/下载:182/47  |  提交时间:2018/05/08
Ra-xii  Cyclopeptide  Autophagy  Apoptosis  Mtor  Hepg2 Liver Cancer Cells  
海棠果降胆固醇药效物质的组学研究 学位论文
: 中国科学院大学, 2017
作者:  文超
Adobe PDF(5378Kb)  |  收藏  |  浏览/下载:173/3  |  提交时间:2019/06/14
Borapetoside E 对高脂饮食诱导小鼠糖脂代谢的影响及其机制研究 学位论文
: 中国科学院大学, 2017
作者:  许宇辉
Adobe PDF(4170Kb)  |  收藏  |  浏览/下载:150/5  |  提交时间:2019/06/14
老药新用:奥柳氮钠的降尿酸作用及分子机制研究 学位论文
: 中国科学院大学, 2017
作者:  牛艳芬
Adobe PDF(4338Kb)  |  收藏  |  浏览/下载:132/6  |  提交时间:2019/06/14
Virtual screening of B-Raf kinase inhibitors: A combination of pharmacophore modelling, molecular docking, 3D-QSAR model and binding free energy calculation studies 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2017, 卷号: 70, 页码: 186-190
作者:  Zhang, Wen;  Qiu, Kai-Xiong;  Yu, Fang;  Xie, Xiao-Guang;  Zhang, Shu-Qun;  Chen, Ya-Juan;  Xie, Hui-Ding
浏览  |  Adobe PDF(371Kb)  |  收藏  |  浏览/下载:171/34  |  提交时间:2017/12/11
B-raf Kinase Inhibitors  Virtual Screening  Pharmacophore  Molecular Docking  3d Qsar  Binding Free Energy Calculation  
Potential role of CYP1B1 in the development and treatment of metabolic diseases 期刊论文
PHARMACOLOGY & THERAPEUTICS, 2017, 卷号: 178, 页码: 18-30
作者:  Li, Fei;  Zhu, Weifeng;  Gonzalez, Frank J.
浏览  |  Adobe PDF(2083Kb)  |  收藏  |  浏览/下载:217/70  |  提交时间:2017/11/20
Cyp1b1  Metabolic Diseases  Metabolic Pathways  Metabolomics  
Using Ultra-Performance Liquid Chromatography Quadrupole Time of Flight Mass Spectrometry-Based Chemometrics for the Identification of Anti-angiogenic Biflavonoids from Edible Garcinia Species 期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2017, 卷号: 65, 期号: 38, 页码: 8348-8355
作者:  Li, Ping;  Yue, Grace Gar-Lee;  Kwok, Hin-Fai;  Long, Chun-lin;  Lau, Clara Bik-San;  Kennelly, Edward J.
浏览  |  Adobe PDF(3340Kb)  |  收藏  |  浏览/下载:372/73  |  提交时间:2017/10/23
Anti-angiogenesis  Garcinia Xanthochymus  Uplc-qtof-ms  Pca  Biflavonoids  
Aspirin increases metabolism through germline signalling to extend the lifespan of Caenorhabditis elegans 期刊论文
PLOS ONE, 2017, 卷号: 12, 期号: 9, 页码: e0184027
作者:  Huang, Xiao-Bing;  Mu, Xiao-Hui;  Wan, Qin-Li;  He, Xiao-Ming;  Wu, Gui-Sheng;  Luo, Huai-Rong
浏览  |  Adobe PDF(7049Kb)  |  收藏  |  浏览/下载:222/43  |  提交时间:2017/10/23
Nonsteroidal Antiinflammatory Drugs  Stem-cells  C. Elegans  Reproductive-system  Sodium-salicylate  Fat-metabolism  Kappa-b  Longevity  Acid  Disease